SCHEMBL4692947

SCHEMBL4692947

Cc1ccc(NCCCN2CC3CN(C(=O)c4ccc(F)cc4F)CC3C2)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPS1 P31327 2/20 0.41
HCRTR1 O43613 2/20 0.41
HCRTR2 O43614 2/20 0.41
KCNK3 O14649 1/20 0.40
KCNK9 Q9NPC2 1/20 0.40
P2RX7 Q99572 2/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
MAPT P10636 3/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 2/20 0.39
HRH1 P35367 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
MAPK14 Q16539 1/20 0.38
GAA P10253 2/20 0.38
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
HTT P42858 1/20 0.38
CCR5 P51681 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694435 0.94 P2RX7 (0.47) HCRTR1HCRTR2KCNK3KCNK9P2RX7
SCHEMBL4692715 0.93 HCRTR1 (0.43) HCRTR1HCRTR2KCNK3KCNK9P2RX7
SCHEMBL4690747 0.93 HCRTR1 (0.41) HCRTR1HCRTR2KCNK3KCNK9P2RX7
SCHEMBL4692704 0.93 HCRTR1 (0.49) HCRTR1HCRTR2KCNK3KCNK9P2RX7
SCHEMBL4693721 0.91 MAPT (0.41) SMN1; SMN2RAB9ANPC1MAPTALDH1A1
SCHEMBL4691905 0.90 HCRTR1 (0.47) HCRTR1HCRTR2KCNK3KCNK9SMN1; SMN2
SCHEMBL4692110 0.89 HCRTR1 (0.51) HCRTR1HCRTR2KCNK3KCNK9P2RX7
SCHEMBL4694970 0.89 LMNA (0.40) HCRTR1HCRTR2KCNK3KCNK9SMN1; SMN2
SCHEMBL4694816 0.89 CCR5 (0.44) HCRTR1HCRTR2SMN1; SMN2RAB9ANPC1
SCHEMBL4695322 0.89 TSHR (0.46) SMN1; SMN2RAB9AMAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed