SCHEMBL4694435

SCHEMBL4694435

Cc1ccc(NCCCN2CC3CN(C(=O)c4ccc(F)cc4Cl)CC3C2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 9/20 0.47
HCRTR1 O43613 1/20 0.42
HCRTR2 O43614 1/20 0.42
HSD11B1 P28845 1/20 0.41
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
AVPR2 P30518 3/20 0.41
KCNK3 O14649 1/20 0.40
KCNK9 Q9NPC2 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
AVPR1A P37288 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692947 0.94 CPS1 (0.41) P2RX7HCRTR1HCRTR2ALDH1A1KCNK3
SCHEMBL4692704 0.93 HCRTR1 (0.49) P2RX7HCRTR1HCRTR2ALDH1A1AVPR2
SCHEMBL4692715 0.92 HCRTR1 (0.43) P2RX7HCRTR1HCRTR2ALDH1A1MEN1
SCHEMBL4690682 0.91 P2RX7 (0.44) P2RX7HCRTR1HCRTR2ALDH1A1AVPR2
SCHEMBL4692110 0.90 HCRTR1 (0.51) P2RX7HCRTR1HCRTR2HSD11B1ALDH1A1
SCHEMBL4692994 0.90 AVPR2 (0.42) ALDH1A1AVPR2NPC1RAB9ASMN1; SMN2
SCHEMBL4695322 0.90 TSHR (0.46) ALDH1A1AVPR2RAB9ASMN1; SMN2MAPT
SCHEMBL4689475 0.89 SMN1; SMN2 (0.39) P2RX7HCRTR1HCRTR2ALDH1A1MEN1
SCHEMBL4694086 0.89 TSHR (0.40) ALDH1A1AVPR2RAB9ASMN1; SMN2MAPT
SCHEMBL4693334 0.89 ALDH1A1 (0.45) P2RX7ALDH1A1KMT2AAVPR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed