SCHEMBL4693100

SCHEMBL4693100

Cc1ccc(NCCCN2CC3CN(C(=O)c4ccc[nH]4)CC3C2)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
MAPT P10636 5/20 0.41
SMN1; SMN2 Q16637 4/20 0.39
GAA P10253 4/20 0.39
KDM4E B2RXH2 1/20 0.39
UBE2M P61081 1/20 0.39
DCUN1D1 Q96GG9 1/20 0.39
HTT P42858 2/20 0.38
LMNA P02545 1/20 0.38
AGTR1 P30556 2/20 0.38
CCR5 P51681 5/20 0.38
RAB9A P51151 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
HRH4 Q9H3N8 1/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695832 0.86 ALDH1A1 (0.38) ALDH1A1MAPTSMN1; SMN2GAAKDM4E
SCHEMBL3281865 0.85 CCR5 (0.52) ALDH1A1MAPTSMN1; SMN2GAAHTT
SCHEMBL4691640 0.85 MAPT (0.54) ALDH1A1MAPTSMN1; SMN2GAAKDM4E
SCHEMBL4693095 0.85 TP53 (0.45) ALDH1A1MAPTSMN1; SMN2GAAKDM4E
SCHEMBL4694532 0.85 DRD3 (0.53) HRH4
SCHEMBL4693334 0.85 ALDH1A1 (0.45) ALDH1A1MAPTSMN1; SMN2GAAKDM4E
SCHEMBL4692889 0.85 MAPT (0.45) ALDH1A1MAPTSMN1; SMN2GAAKDM4E
SCHEMBL4693486 0.84 HCRTR1 (0.48) ALDH1A1MAPTSMN1; SMN2GAAKDM4E
SCHEMBL4694235 0.84 ALDH1A1 (0.43) ALDH1A1MAPTSMN1; SMN2GAAKDM4E
SCHEMBL14436612 0.84 ALDH1A1 (0.45) ALDH1A1MAPTSMN1; SMN2GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed