SCHEMBL4693170

SCHEMBL4693170

Cc1ccc(NCCCN2CC3CN(C(=O)c4cc(F)ccc4C(F)(F)F)CC3C2)cc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 5/20 0.51
HCRTR2 O43614 5/20 0.51
SCD O00767 1/20 0.40
KCNK3 O14649 1/20 0.40
KCNK9 Q9NPC2 1/20 0.40
RAF1 P04049 1/20 0.39
ARAF P10398 1/20 0.39
BRAF P15056 1/20 0.39
P2RX7 Q99572 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ALDH1A1 P00352 4/20 0.37
MAPT P10636 4/20 0.37
HTT P42858 2/20 0.37
NPY2R P49146 1/20 0.37
GRIN2B Q13224 1/20 0.37
USP2 O75604 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692110 0.93 HCRTR1 (0.51) HCRTR1HCRTR2SCDKCNK3KCNK9
SCHEMBL4692704 0.91 HCRTR1 (0.49) HCRTR1HCRTR2KCNK3KCNK9P2RX7
SCHEMBL4693018 0.90 NPY2R (0.47) SCDSMN1; SMN2ALDH1A1MAPTNPY2R
SCHEMBL4692715 0.89 HCRTR1 (0.43) HCRTR1HCRTR2KCNK3KCNK9P2RX7
SCHEMBL4694435 0.88 P2RX7 (0.47) HCRTR1HCRTR2KCNK3KCNK9P2RX7
SCHEMBL4695365 0.88 BRAF (0.39) HCRTR1HCRTR2RAF1ARAFBRAF
SCHEMBL4692947 0.88 CPS1 (0.41) HCRTR1HCRTR2KCNK3KCNK9P2RX7
SCHEMBL4693167 0.87 HCRTR1 (0.50) HCRTR1HCRTR2SMN1; SMN2NPC1RAB9A
SCHEMBL4691185 0.87 P2RX7 (0.43) HCRTR1HCRTR2RAF1ARAFBRAF
SCHEMBL4690182 0.86 RBP4 (0.41) HCRTR1HCRTR2RAF1ARAFBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed