SCHEMBL4693214

SCHEMBL4693214

COc1ccc(COc2ccc(C(=O)NCC(C)O)cc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.67
MAPT P10636 3/20 0.67
HTT P42858 1/20 0.67
SMN1; SMN2 Q16637 4/20 0.59
NPC1 O15118 4/20 0.59
RAB9A P51151 4/20 0.59
POLB P06746 1/20 0.59
GAA P10253 1/20 0.55
KMT2A Q03164 5/20 0.55
MEN1 O00255 3/20 0.55
ADAM17 P78536 1/20 0.55
FFAR1 O14842 1/20 0.54
HPGD P15428 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
PLA2G4B P0C869 1/20 0.53
MAPK1 P28482 1/20 0.52
EPHX2 P34913 1/20 0.50
NR1H4 Q96RI1 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
LMNA P02545 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5856056 0.89 ALDH1A1 (0.68) ALDH1A1SMN1; SMN2NPC1RAB9AGAA
SCHEMBL4693371 0.81 ALDH1A1 (0.70) ALDH1A1MAPTHTTSMN1; SMN2NPC1
SCHEMBL3201438 0.80 ALDH1A1 (1.00) ALDH1A1MAPTHTTSMN1; SMN2NPC1
SCHEMBL4754917 0.80 ALDH1A1 (0.78) ALDH1A1MAPTHTTSMN1; SMN2NPC1
SCHEMBL3729907 0.80 NPC1 (0.75) ALDH1A1MAPTHTTSMN1; SMN2NPC1
SCHEMBL3604393 0.79 SMN1; SMN2 (0.68) ALDH1A1MAPTHTTSMN1; SMN2NPC1
SCHEMBL3604397 0.79 SMN1; SMN2 (0.68) ALDH1A1MAPTHTTSMN1; SMN2NPC1
SCHEMBL5641504 0.79 ADRB2 (0.68) ALDH1A1MAPTHTTSMN1; SMN2NPC1
SCHEMBL24225548 0.78 HPGD (0.71) ALDH1A1SMN1; SMN2NPC1RAB9AGAA
SCHEMBL22386732 0.77 SMN1; SMN2 (0.69) ALDH1A1MAPTHTTSMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1521757-B1 TRICYCLIC SPIROPIPERIDINES OR SPIROPYRROLIDINES ASTRAZENECA AB (SE) 2008-01-30 EP disclosed