SCHEMBL4693239

SCHEMBL4693239

Cc1cccc(CC(N)C(C)C)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 6/20 0.50
IDO1 P14902 2/20 0.48
PNMT P11086 1/20 0.47
SLC6A2 P23975 2/20 0.45
MAOA P21397 1/20 0.45
SLC6A4 P31645 1/20 0.45
SLC6A3 Q01959 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
CYP2A6 P11509 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43
HTR2B P41595 2/20 0.43
ALDH1A1 P00352 1/20 0.41
CYP2D6 P10635 1/20 0.41
ACHE P22303 1/20 0.41
SCN4A P35499 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29968153 0.86 PNMT (0.62) TAAR1IDO1PNMTSLC6A2MAOA
SCHEMBL2563917 0.86 PNMT (0.62) TAAR1IDO1PNMTSLC6A2MAOA
SCHEMBL12136140 0.86 PNMT (0.62) TAAR1IDO1PNMTSLC6A2MAOA
SCHEMBL10249345 0.86 PNMT (0.62) TAAR1IDO1PNMTSLC6A2MAOA
Hydrochloric Acid SCHEMBL30559539 0.84 PNMT (0.60) TAAR1IDO1PNMTSLC6A2MAOA
SCHEMBL7694750 0.82 TAAR1 (0.55) TAAR1IDO1PNMTSLC6A2MAOA
SCHEMBL6170324 0.80 TAAR1 (0.46) TAAR1IDO1PNMTSLC6A2MAOA
SCHEMBL598282 0.79 TAAR1 (0.52) TAAR1IDO1PNMTSLC6A2MAOA
SCHEMBL3126846 0.79 TAAR1 (0.48) TAAR1IDO1PNMTSLC6A2MAOA
SCHEMBL4692874 0.79 ADRB1 (0.53) TAAR1PNMTSLC6A2MAOASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1375489-B1 MEDICINAL COMPOSITION CONTAINING 1,3-THIAZINE DERIVATIVE SHIONOGI & CO (JP) 2008-08-20 EP disclosed
US-6916806-B2 Medicinal composition containing 1,3-thiazine derivative SHIONOGI & CO., LTD. (JP) 2005-07-12 US disclosed
US-20040116326-A1 Medicinal composition containing 1,3-thiazine derivative SHIONOGI & CO., LTD. (JP) 2004-06-17 US disclosed
EP-1375489-A1 MEDICINAL COMPOSITION CONTAINING 1,3-THIAZINE DERIVATIVE SHIONOGI & CO., LTD. (JP) 2004-01-02 EP disclosed