SCHEMBL4695600

SCHEMBL4695600

O=C(O)C1c2c(cnn2-c2ccccc2)C(NOCc2ccccc2)CN1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
LMNA P02545 2/20 0.37
SLC9A1 P19634 1/20 0.35
SLC9A2 Q9UBY0 1/20 0.35
KMT2A Q03164 2/20 0.35
HTT P42858 1/20 0.35
MAPK14 Q16539 1/20 0.35
HPGD P15428 1/20 0.34
NPC1 O15118 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
RAB9A P51151 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
TP53 P04637 2/20 0.33
ACHE P22303 1/20 0.33
MAPT P10636 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4138926 0.91 KEAP1 (0.38) KEAP1NFE2L2LMNASLC9A1SLC9A2
SCHEMBL3305431 0.87 LMNA (0.34) LMNANPC1RAB9AACHE
SCHEMBL5254943 0.80 NPC1 (0.38) NPC1MAPK1RAB9A
SCHEMBL4693843 0.80 KEAP1 (0.40) KEAP1NFE2L2LMNASLC9A1SLC9A2
SCHEMBL4695496 0.78 KEAP1 (0.45) KEAP1NFE2L2SLC9A1SLC9A2KMT2A
Hydrochloric Acid SCHEMBL4145877 0.75 HTT (0.39) KEAP1NFE2L2LMNAKMT2AHTT
SCHEMBL4697074 0.74 NPC1 (0.34) NPC1RAB9A
SCHEMBL5187275 0.73 GPR183 (0.39) HPGDNPC1TSHRRAB9ATDP1
SCHEMBL4697059 0.71 AGTR2 (0.32) NPC1RAB9A
SCHEMBL4147781 0.71 KEAP1 (0.41) KEAP1NFE2L2SLC9A1SLC9A2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569935-B1 HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREOF AND USE OF SAME AS MEDICAMENTS, SUCH AS ANTI-BACTERIAL MEDICAMENTS AND BETA-LACTAMASE INHIBITORS NOVEXEL (FR) 2008-08-20 EP disclosed