SCHEMBL4693907

SCHEMBL4693907

Cc1ccc(C(CC(N)=O)N2CC3CN(C(=O)c4ccccc4C#N)CC3C2)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 6/20 0.48
HCRTR2 O43614 6/20 0.48
TNF P01375 2/20 0.40
PDE2A O00408 1/20 0.36
HSD11B1 P28845 1/20 0.36
KDM1A O60341 1/20 0.36
CYP2C9 P11712 2/20 0.34
CYP2D6 P10635 1/20 0.34
SLC9A1 P19634 1/20 0.34
CYP2C19 P33261 1/20 0.34
MGLL Q99685 1/20 0.34
RORC P51449 1/20 0.34
PGR P06401 2/20 0.33
GBA1 P04062 1/20 0.33
CCL5 P13501 1/20 0.33
CCR5 P51681 1/20 0.33
KCNK3 O14649 1/20 0.33
KCNK9 Q9NPC2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692886 0.89 ALDH1A1 (0.42) HCRTR1HCRTR2TNFCYP2C9CYP2C19
SCHEMBL4694224 0.86 TNF (0.39) HCRTR1HCRTR2TNFMGLLGBA1
SCHEMBL4693484 0.86 HCRTR1 (0.48) HCRTR1HCRTR2TNFGBA1CCR5
SCHEMBL4691904 0.86 HCRTR1 (0.46) HCRTR1HCRTR2TNFKCNK3KCNK9
SCHEMBL4691868 0.85 HCRTR1 (0.47) HCRTR1HCRTR2TNFGBA1CCR5
SCHEMBL4694354 0.85 P2RX7 (0.44) HCRTR1HCRTR2TNF
SCHEMBL4690634 0.85 TNF (0.38) HCRTR1HCRTR2TNFGBA1CCR5
SCHEMBL4691405 0.85 HCRTR1 (0.48) HCRTR1HCRTR2TNFCYP2C9CYP2C19
SCHEMBL4694616 0.85 TNF (0.38) HCRTR1HCRTR2TNFGBA1CCR5
SCHEMBL4696301 0.84 LMNA (0.42) HCRTR1HCRTR2TNFSLC9A1GBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed