SCHEMBL4694247

SCHEMBL4694247

Cc1c(S(=O)(=O)N2CC3CN(CC[C@H](N)c4ccccc4)CC3C2)cnn1-c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
SMO Q99835 1/20 0.36
CCKBR P32239 1/20 0.35
CCL5 P13501 7/20 0.35
MAPK1 P28482 1/20 0.35
MAPT P10636 2/20 0.34
CCR5 P51681 4/20 0.34
SLC9A1 P19634 1/20 0.34
SLC9A2 Q9UBY0 1/20 0.34
ALDH1A1 P00352 1/20 0.34
APP P05067 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3282872 1.00 DRD2 (0.36) DRD2DRD4DRD3SMOCCKBR
Cyclopentane SCHEMBL4691240 0.83 CCR5 (0.48) MAPK1CCR5
SCHEMBL4690865 0.81 CCR5 (0.46) CCL5MAPK1MAPTCCR5SLC9A1
SCHEMBL13326752 0.79 CCR5 (0.61) CCR5
SCHEMBL5421969 0.79 CCR5 (0.61) CCR5
SCHEMBL4694250 0.77 CCR5 (0.44) CCL5MAPK1MAPTCCR5ALDH1A1
SCHEMBL4692842 0.76 GBA1 (0.43) CCR5ALDH1A1
SCHEMBL4691491 0.75 FPR2 (0.50) ALDH1A1
SCHEMBL4693317 0.75 EIF4A3 (0.49) CCL5MAPK1MAPTCCR5ALDH1A1
SCHEMBL4690883 0.75 NR1H4 (0.41) MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed