SCHEMBL4694350

SCHEMBL4694350

COc1ccc(F)cc1C(=O)N1CC2CN(C(CC(N)=O)c3ccc(C)c(Cl)c3)CC2C1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 2/20 0.42
KCNK9 Q9NPC2 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
HCRTR1 O43613 6/20 0.40
HCRTR2 O43614 6/20 0.40
PDE2A O00408 1/20 0.38
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
TNF P01375 1/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
P2RX7 Q99572 1/20 0.37
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692703 0.91 HCRTR1 (0.48) KCNK3KCNK9HCRTR1HCRTR2PDE2A
SCHEMBL4691836 0.91 HCRTR2 (0.40) SMN1; SMN2HCRTR1HCRTR2PDE4APDE4B
SCHEMBL4691405 0.91 HCRTR1 (0.48) KCNK3KCNK9HCRTR1HCRTR2PDE4A
SCHEMBL4692712 0.90 HCRTR1 (0.43) KCNK3KCNK9HCRTR1HCRTR2TNF
SCHEMBL4693952 0.88 HCRTR1 (0.50) HCRTR1HCRTR2PDE2APDE4APDE4B
SCHEMBL4692944 0.88 HCRTR1 (0.41) KCNK3KCNK9SMN1; SMN2HCRTR1HCRTR2
SCHEMBL4693169 0.86 HCRTR1 (0.50) KCNK3KCNK9HCRTR1HCRTR2P2RX7
SCHEMBL4692627 0.86 HCRTR1 (0.50) SMN1; SMN2HCRTR1HCRTR2ALDH1A1KDM4E
SCHEMBL4693896 0.86 HCRTR1 (0.47) SMN1; SMN2HCRTR1HCRTR2PDE4APDE4B
SCHEMBL4694424 0.85 HCRTR1 (0.37) HCRTR1HCRTR2PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed