SCHEMBL4694424

SCHEMBL4694424

COc1cscc1C(=O)N1CC2CN(C(CC(N)=O)c3ccc(C)c(Cl)c3)CC2C1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 12/20 0.37
HCRTR2 O43614 12/20 0.37
TNF P01375 4/20 0.36
PDE4A P27815 3/20 0.36
PDE4B Q07343 3/20 0.36
PDE4C Q08493 3/20 0.36
PDE4D Q08499 3/20 0.36
HTR1A P08908 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691405 0.88 HCRTR1 (0.48) HCRTR1HCRTR2TNFPDE4APDE4B
SCHEMBL4693952 0.87 HCRTR1 (0.50) HCRTR1HCRTR2TNFPDE4APDE4B
SCHEMBL4695901 0.86 HCRTR2 (0.47) HCRTR1HCRTR2
SCHEMBL4691836 0.86 HCRTR2 (0.40) HCRTR1HCRTR2TNFPDE4APDE4B
SCHEMBL4692627 0.85 HCRTR1 (0.50) HCRTR1HCRTR2
SCHEMBL4694350 0.85 KCNK3 (0.42) HCRTR1HCRTR2TNFPDE4APDE4B
SCHEMBL4693896 0.85 HCRTR1 (0.47) HCRTR1HCRTR2TNFPDE4APDE4B
SCHEMBL4690309 0.84 HCRTR1 (0.38) HCRTR1HCRTR2TNFPDE4APDE4B
SCHEMBL4691302 0.84 HCRTR1 (0.42) HCRTR1HCRTR2TNFPDE4APDE4B
SCHEMBL4690927 0.84 HCRTR1 (0.49) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed