SCHEMBL4693952

SCHEMBL4693952

COc1cccc(C(=O)N2CC3CN(C(CC(N)=O)c4ccc(C)c(Cl)c4)CC3C2)c1C

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 11/20 0.50
HCRTR2 O43614 11/20 0.50
PDE4A P27815 2/20 0.39
PDE4B Q07343 2/20 0.39
PDE4C Q08493 2/20 0.39
PDE4D Q08499 2/20 0.39
TNF P01375 1/20 0.39
UTS2R Q9UKP6 2/20 0.37
PDE2A O00408 1/20 0.37
MGLL Q99685 1/20 0.37
POLB P06746 1/20 0.37
NPC1 O15118 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691405 0.94 HCRTR1 (0.48) HCRTR1HCRTR2PDE4APDE4BPDE4C
SCHEMBL4692627 0.93 HCRTR1 (0.50) HCRTR1HCRTR2POLBNPC1
SCHEMBL4693896 0.91 HCRTR1 (0.47) HCRTR1HCRTR2PDE4APDE4BPDE4C
SCHEMBL4691868 0.91 HCRTR1 (0.47) HCRTR1HCRTR2TNF
SCHEMBL4691302 0.90 HCRTR1 (0.42) HCRTR1HCRTR2PDE4APDE4BPDE4C
SCHEMBL4695647 0.89 HCRTR1 (0.48) HCRTR1HCRTR2TNFPDE2A
SCHEMBL4694350 0.88 KCNK3 (0.42) HCRTR1HCRTR2PDE4APDE4BPDE4C
SCHEMBL4694354 0.87 P2RX7 (0.44) HCRTR1HCRTR2TNF
SCHEMBL4692886 0.87 ALDH1A1 (0.42) HCRTR1HCRTR2TNFMGLL
SCHEMBL4694424 0.87 HCRTR1 (0.37) HCRTR1HCRTR2PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed