SCHEMBL4690682

SCHEMBL4690682

Cc1ccc(NCCCN2CC3CN(C(=O)c4ccc(Cl)cc4Cl)CC3C2)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.44
HCRTR1 O43613 2/20 0.42
HCRTR2 O43614 2/20 0.42
AVPR2 P30518 4/20 0.41
MAPT P10636 3/20 0.40
ALDH1A1 P00352 3/20 0.40
UBE2M P61081 1/20 0.40
DCUN1D1 Q96GG9 1/20 0.40
FLT1 P17948 1/20 0.39
FLT4 P35916 1/20 0.39
KDR P35968 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 2/20 0.39
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690670 0.94 UBE2M (0.44) HCRTR1HCRTR2AVPR2MAPTALDH1A1
SCHEMBL4694270 0.93 HCRTR1 (0.50) HCRTR1HCRTR2MAPTALDH1A1UBE2M
SCHEMBL4690747 0.93 HCRTR1 (0.41) P2RX7HCRTR1HCRTR2MAPTALDH1A1
SCHEMBL4692694 0.92 LMNA (0.46) HCRTR1HCRTR2MAPTALDH1A1UBE2M
SCHEMBL4694435 0.91 P2RX7 (0.47) P2RX7HCRTR1HCRTR2AVPR2MAPT
SCHEMBL4692994 0.91 AVPR2 (0.42) AVPR2MAPTALDH1A1UBE2MDCUN1D1
SCHEMBL4690506 0.90 HCRTR1 (0.52) HCRTR1HCRTR2MAPTALDH1A1LMNA
SCHEMBL4693334 0.89 ALDH1A1 (0.45) P2RX7AVPR2MAPTALDH1A1UBE2M
SCHEMBL4691668 0.89 GPR6 (0.42) AVPR2MAPTALDH1A1SMN1; SMN2LMNA
SCHEMBL4694970 0.89 LMNA (0.40) HCRTR1HCRTR2AVPR2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed