SCHEMBL4694469

SCHEMBL4694469

COc1ccc2[nH]c(C)c(CC(=O)OCC(=O)OC(C)(C)C)c2c1C(=O)c1ccc(Cl)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.37
KLK6 Q92876 2/20 0.35
HTR1A P08908 1/20 0.35
PKM P14618 1/20 0.35
PTGS1 P23219 1/20 0.35
GLO1 Q04760 1/20 0.35
HIF1A Q16665 1/20 0.35
POLB P06746 2/20 0.35
PRSS1 P07477 1/20 0.35
PRSS2 P07478 1/20 0.35
PRSS3 P35030 1/20 0.35
HPGD P15428 2/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAPT P10636 2/20 0.34
PTGDR Q13258 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
LMNA P02545 1/20 0.33
CNR1 P21554 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691290 0.89 PTGS1 (0.44) PTGS2KLK6HTR1APKMPTGS1
SCHEMBL7761162 0.84 PTGS2 (0.39) PTGS2POLBHPGDTP53SMN1; SMN2
SCHEMBL998208 0.83 AKR1C2 (0.46) PTGS2PTGS1GLO1HIF1APOLB
SCHEMBL5154201 0.83 POLB (0.41) PKMPOLBHPGDMAPTPTGDR
SCHEMBL4695816 0.80 PTGS2 (0.42) PTGS2KLK6PTGS1POLBPRSS1
SCHEMBL5154300 0.79 POLB (0.38) PTGS2POLBHPGDMAPTPTGDR
SCHEMBL18765238 0.79 POLB (0.38) PTGS2PTGS1POLBHPGDMAPT
SCHEMBL4692036 0.79 PTGS2 (0.34) PTGS2KLK6HTR1APKMPTGS1
SCHEMBL5806535 0.79 POLB (0.41) PTGS1POLBHPGDMAPTLMNA
SCHEMBL6589711 0.79 MEN1 (0.37) PTGS2PTGS1POLBHPGDTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539729-A4 NITROSATED NONSTEROIDAL ANTIINFLAMMATORY COMPOUNDS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-02-20 EP disclosed
EP-1539729-A2 NITROSATED NONSTEROIDAL ANTIINFLAMMATORY COMPOUNDS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-15 EP disclosed
WO-2004004648-A2 NITROSATED NONSTEROIDAL ANTIINFLAMMATORY COMPOUNDS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-15 WO disclosed