SCHEMBL5806535

SCHEMBL5806535

COc1ccc2[nH]c(C)c(CCO)c2c1C(=O)c1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.41
MAPT P10636 3/20 0.40
CYP2C9 P11712 1/20 0.40
PTGS1 P23219 1/20 0.39
HPGD P15428 1/20 0.39
CNR1 P21554 1/20 0.38
GAA P10253 2/20 0.37
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
SLC2A1 P11166 1/20 0.36
LMNA P02545 2/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
TACR1 P25103 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5805761 0.89 KRAS (0.43) POLBMAPTCYP2C9HPGDCNR1
SCHEMBL8889810 0.88 POLB (0.39) POLBMAPTCYP2C9HPGDCNR1
SCHEMBL5805796 0.87 POLB (0.40) POLBMAPTHPGDCNR1GAA
SCHEMBL998208 0.86 AKR1C2 (0.46) POLBMAPTCYP2C9PTGS1HPGD
SCHEMBL5154201 0.86 POLB (0.41) POLBMAPTHPGDCNR1GAA
SCHEMBL8671570 0.85 POLB (0.40) POLBMAPTPTGS1HPGDCNR1
SCHEMBL5805625 0.85 PTGS2 (0.38) POLBMAPTPTGS1HPGDCNR1
SCHEMBL5808478 0.84 PTGS1 (0.49) POLBMAPTCYP2C9PTGS1HPGD
SCHEMBL7761162 0.84 PTGS2 (0.39) POLBMAPTHPGDCNR1TSHR
SCHEMBL8646568 0.84 ALDH1A1 (0.40) POLBMAPTHPGDGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006099416-A1 2-METHYL INDOLE CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2006-09-21 WO claimed
WO-2006099416-A1 2-METHYL INDOLE CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2006-09-21 WO disclosed
US-5756531-A ANTIALLERGENS; ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES (US) 1998-05-26 US disclosed
US-5750558-A ANTIALLERGENS, ANTIINFLAMMATORY AGENTS ABBOTT LABORATORIES (US) 1998-05-12 US disclosed
WO-1997041100-A1 IMINOXY DERIVATIVES OF INDOLE AND INDENE COMPOUNDS AS INHIBITORS OF PROSTAGLANDIN BIOSYNTHESIS ABBOTT LABORATORIES (US) 1997-11-06 WO disclosed