SCHEMBL4694867

SCHEMBL4694867

Cc1ccc(N(CCCN2CC3=CN(C(=O)c4c(C)ccnc4C)CC3C2)C(=O)Nc2ccc(Cl)cc2C(F)(F)F)cc1Cl

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 10/20 0.34
KCNH2 Q12809 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
PROKR1 Q8TCW9 5/20 0.33
TP53 P04637 2/20 0.31
MAPT P10636 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694359 0.92 CCR5 (0.34) CCR5KCNH2
SCHEMBL4753854 0.89 CCR5 (0.34) CCR5KCNH2
SCHEMBL4690445 0.88 EPHX2 (0.38) CCR5KCNH2
SCHEMBL4690306 0.88 CCR5 (0.38) CCR5KCNH2TRPV1
SCHEMBL4691638 0.86 CCR5 (0.37) CCR5KCNH2
SCHEMBL4691722 0.86 CCR5 (0.39) CCR5KCNH2TP53MAPTSMN1; SMN2
SCHEMBL4694864 0.86 CCR5 (0.40) CCR5KCNH2TRPV1PROKR1TP53
SCHEMBL4690740 0.86 CCR5 (0.42) CCR5KCNH2
SCHEMBL4690611 0.85 CCR5 (0.37) CCR5KCNH2MAPT
SCHEMBL4694952 0.85 CCR5 (0.37) CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed