SCHEMBL4694978

SCHEMBL4694978

N#Cc1cccc(C(=O)N[C@@H](CCN2CC3=CN(C(=O)c4c(F)cccc4Cl)CC3C2)c2ccccc2)c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 6/20 0.41
UTS2R Q9UKP6 4/20 0.39
S1PR3 Q99500 3/20 0.37
S1PR4 O95977 1/20 0.37
GPR139 Q6DWJ6 1/20 0.37
DGAT2 Q96PD7 1/20 0.37
DRD4 P21917 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
RORC P51449 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694186 0.93 CCR5 (0.42) CCR5UTS2RDGAT2
SCHEMBL4691249 0.92 CCR5 (0.44) CCR5UTS2RGPR139DGAT2
SCHEMBL4690858 0.92 CCR5 (0.48) CCR5UTS2RDGAT2
SCHEMBL4696133 0.90 CCR5 (0.46) CCR5UTS2RDGAT2
SCHEMBL4692159 0.89 CCR5 (0.42) CCR5UTS2RDGAT2
SCHEMBL4694054 0.89 CCR5 (0.42) CCR5UTS2RDGAT2DRD4
SCHEMBL4690242 0.89 CCR5 (0.43) CCR5UTS2RDGAT2
SCHEMBL4692359 0.89 CCR5 (0.42) CCR5UTS2RGPR139DRD4
SCHEMBL4690226 0.88 CCR5 (0.46) CCR5UTS2R
SCHEMBL4695516 0.88 CCR5 (0.41) CCR5UTS2RGPR139DGAT2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed