SCHEMBL4692359

SCHEMBL4692359

COc1cccc(C(=O)N[C@@H](CCN2CC3=CN(C(=O)c4c(F)cccc4Cl)CC3C2)c2ccccc2)c1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 4/20 0.42
ROCK2 O75116 2/20 0.42
ROCK1 Q13464 2/20 0.42
DRD4 P21917 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
MAPK1 P28482 1/20 0.41
KMT2A Q03164 1/20 0.41
UTS2R Q9UKP6 2/20 0.39
GPR139 Q6DWJ6 4/20 0.39
CTSS P25774 1/20 0.39
DRD2 P14416 1/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691378 0.93 CCR5 (0.43) CCR5ROCK2ROCK1ALDH1A1MEN1
SCHEMBL4691249 0.91 CCR5 (0.44) CCR5ROCK2ROCK1KMT2AUTS2R
SCHEMBL4690858 0.91 CCR5 (0.48) CCR5ROCK2ROCK1UTS2R
SCHEMBL4691873 0.91 ACHE (0.45) CCR5ROCK2ROCK1DRD4ALDH1A1
SCHEMBL4696133 0.90 CCR5 (0.46) CCR5UTS2RLMNAGAA
SCHEMBL4694978 0.89 CCR5 (0.41) CCR5DRD4UTS2RGPR139
SCHEMBL4692159 0.89 CCR5 (0.42) CCR5ROCK2ROCK1MEN1KMT2A
SCHEMBL4694054 0.89 CCR5 (0.42) CCR5ROCK2ROCK1DRD4UTS2R
SCHEMBL4690242 0.89 CCR5 (0.43) CCR5ROCK2ROCK1UTS2R
SCHEMBL4691824 0.88 CCR5 (0.42) CCR5MEN1KMT2AUTS2RLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed