SCHEMBL4695205

SCHEMBL4695205

CS(=O)(=O)c1cc2c[c]ccc2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CA2 P00918 7/20 0.40
CNR1 P21554 6/20 0.35
PTGS2 P35354 1/20 0.32
AKR1B1 P15121 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL694332 0.77 CA2 (0.42) CA2CNR1AKR1B1
SCHEMBL7014167 0.76 CA2 (0.67) CA2CNR1AKR1B1
SCHEMBL445877 0.71 CYP2A6 (0.48) PTGS2
SCHEMBL7372883 0.69 BRD4 (0.59)
SCHEMBL7758397 0.68 FLT3 (0.42)
SCHEMBL4467591 0.67
SCHEMBL4717754 0.67 AOC3 (0.54)
SCHEMBL2452605 0.67 DAO (0.31)
SCHEMBL4460967 0.67 F11 (0.31)
SCHEMBL8205395 0.67 CYP2A6 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960355-A1 3-AMINO-1-ARYLPROPYL INDOLES AND AZA-SUBSTITUTED INDOLES F.HOFFMANN-LA ROCHE AG (CH) 2008-08-27 EP disclosed
WO-2007062996-A1 3-AMINO-1-ARYLPROPYL INDOLES AND AZA-SUBSTITUTED INDOLES F. HOFFMANN-LA ROCHE AG (CH) 2007-06-07 WO disclosed