SCHEMBL4695787

SCHEMBL4695787

Cc1ccc(NC(=O)CCN2CC3CNCC3[C@H]2C(=O)c2cccnc2N(C)C)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.39
MALT1 Q9UDY8 1/20 0.38
MAPT P10636 5/20 0.38
LMNA P02545 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 2/20 0.37
GBA1 P04062 1/20 0.37
HTT P42858 1/20 0.37
GAA P10253 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
POLB P06746 1/20 0.36
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
THRB P10828 1/20 0.36
DRD2 P14416 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4696289 0.83 THRB (0.38) TP53MALT1MAPTLMNAALDH1A1
SCHEMBL4695194 0.79 TP53 (0.42) TP53MALT1MAPTLMNAMEN1
SCHEMBL4695896 0.78 POLB (0.46) TP53MAPTMEN1KMT2AALDH1A1
SCHEMBL4694793 0.77 MAPT (0.43) TP53MAPTLMNAMEN1KMT2A
SCHEMBL3286924 0.74 TP53 (0.53) TP53MAPTLMNAMEN1KMT2A
SCHEMBL4690604 0.71 TP53 (0.44) TP53MALT1MAPTLMNAMEN1
SCHEMBL4690539 0.70 TP53 (0.45) TP53MALT1MAPTLMNAMEN1
SCHEMBL4695171 0.69 TP53 (0.40) TP53MAPTLMNAMEN1KMT2A
SCHEMBL3283676 0.68 TP53 (0.53) TP53MALT1MAPTLMNAMEN1
SCHEMBL5662686 0.68 MALT1 (0.50) TP53MALT1MAPTALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed