SCHEMBL4696289

SCHEMBL4696289

Cc1ccc(NC(=O)CCN2CC3CNCC3[C@H]2C(=O)c2c(C)ccnc2C)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.38
LMNA P02545 3/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 3/20 0.38
MALT1 Q9UDY8 1/20 0.38
NPC1 O15118 1/20 0.38
GAA P10253 1/20 0.38
RAB9A P51151 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695787 0.83 TP53 (0.39) THRBLMNATP53MAPTMALT1
SCHEMBL4695896 0.80 POLB (0.46) THRBTP53MAPTNPC1RAB9A
SCHEMBL4694793 0.79 MAPT (0.43) THRBLMNATP53MAPTNPC1
SCHEMBL3282221 0.78 CCR5 (0.51) LMNATP53MAPTALDH1A1GLA
SCHEMBL3286924 0.77 TP53 (0.53) LMNATP53MAPTALDH1A1CYP2C9
SCHEMBL4747293 0.75 CCR5 (0.36) RAB9A
SCHEMBL4693617 0.72 CCR5 (0.51) LMNAMAPTALDH1A1MAPK1
SCHEMBL3285287 0.72 TP53 (0.43) LMNATP53MAPTRAB9AALDH1A1
SCHEMBL3283571 0.71 CCR5 (0.44) THRBLMNATP53MAPTALDH1A1
SCHEMBL4695429 0.70 CCR5 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed