SCHEMBL4695977

SCHEMBL4695977

O=C(c1ccc(-c2ccccc2F)cc1C(F)(F)F)N1CCN(c2ncccn2)CC1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A7 Q99884 9/20 0.62
KDM4E B2RXH2 3/20 0.62
ALDH1A1 P00352 3/20 0.62
L3MBTL1 Q9Y468 2/20 0.62
TSHR P16473 1/20 0.49
SCD O00767 1/20 0.48
DRD2 P14416 1/20 0.48
DRD4 P21917 1/20 0.48
DRD3 P35462 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPK1 P28482 1/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3817716 0.87 SLC6A7 (0.63) SLC6A7KDM4EALDH1A1L3MBTL1TSHR
SCHEMBL3821678 0.85 ALDH1A1 (0.65) SLC6A7KDM4EALDH1A1L3MBTL1TSHR
SCHEMBL5935798 0.83 SLC6A7 (0.59) SLC6A7KDM4EALDH1A1L3MBTL1TSHR
SCHEMBL4699807 0.82 SLC6A7 (0.46) SLC6A7KDM4EALDH1A1L3MBTL1DRD2
SCHEMBL3821810 0.80 SLC6A7 (0.44) SLC6A7KDM4EALDH1A1L3MBTL1TSHR
SCHEMBL3578554 0.77 SLC6A7 (1.00) SLC6A7ALDH1A1L3MBTL1TSHR
SCHEMBL3578419 0.77 SLC6A7 (0.77) SLC6A7KDM4EALDH1A1L3MBTL1TSHR
SCHEMBL3817981 0.77 ALDH1A1 (0.64) SLC6A7KDM4EALDH1A1L3MBTL1TSHR
SCHEMBL3580180 0.75 KDM4E (0.71) SLC6A7KDM4EALDH1A1L3MBTL1TSHR
SCHEMBL3413095 0.74 P2RX7 (0.62) KDM4EALDH1A1TSHRSCDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893212-A2 MULTICYCLIC COMPOUNDS AND METHODS OF THEIR USE Lexicon Pharmaceuticals, Inc. (US) 2008-03-05 EP claimed
WO-2006124748-A2 MULTICYCLIC COMPOUNDS AND METHODS OF THEIR USE LEXICON GENETICS INCORPORATED (US) 2006-11-23 WO claimed
EP-1893212-A2 MULTICYCLIC COMPOUNDS AND METHODS OF THEIR USE Lexicon Pharmaceuticals, Inc. (US) 2008-03-05 EP disclosed
WO-2006124748-A2 MULTICYCLIC COMPOUNDS AND METHODS OF THEIR USE LEXICON GENETICS INCORPORATED (US) 2006-11-23 WO disclosed