SCHEMBL4699807

SCHEMBL4699807

CC1(C(=O)c2ccc(-c3ccccc3F)cc2C(F)(F)F)CCN(c2ncccn2)CC1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A7 Q99884 5/20 0.46
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
WDR5 P61964 6/20 0.41
CYP2C9 P11712 2/20 0.39
USP2 O75604 1/20 0.39
MAPK1 P28482 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695977 0.82 SLC6A7 (0.62) SLC6A7DRD2DRD4DRD3KDM4E
SCHEMBL3821810 0.77 SLC6A7 (0.44) SLC6A7DRD2DRD4DRD3KDM4E
SCHEMBL3584830 0.76 SLC6A7 (0.50) SLC6A7L3MBTL1CYP2C9USP2CYP1A2
SCHEMBL3821678 0.69 ALDH1A1 (0.65) SLC6A7DRD2DRD4DRD3KDM4E
SCHEMBL3817716 0.69 SLC6A7 (0.63) SLC6A7KDM4EALDH1A1L3MBTL1
SCHEMBL5935798 0.66 SLC6A7 (0.59) SLC6A7KDM4EALDH1A1L3MBTL1
SCHEMBL15416474 0.64 MEN1 (0.58) KDM4EALDH1A1CYP2C9USP2MAPK1
SCHEMBL3815687 0.64 MALT1 (0.48) SLC6A7KDM4EL3MBTL1CYP2C19MEN1
SCHEMBL3578554 0.63 SLC6A7 (1.00) SLC6A7ALDH1A1L3MBTL1
SCHEMBL3580180 0.62 KDM4E (0.71) SLC6A7KDM4EALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893212-A2 MULTICYCLIC COMPOUNDS AND METHODS OF THEIR USE Lexicon Pharmaceuticals, Inc. (US) 2008-03-05 EP claimed
WO-2006124748-A2 MULTICYCLIC COMPOUNDS AND METHODS OF THEIR USE LEXICON GENETICS INCORPORATED (US) 2006-11-23 WO claimed
WO-2006124897-A2 METHODS AND COMPOSITIONS FOR IMPROVING COGNITION LEXICON GENETICS INCORPORATED (US) 2006-11-23 WO disclosed