SCHEMBL4696795

SCHEMBL4696795

CN(CCOC(=O)N(c1ccccc1-c1ccccc1)N1CC[CH]CC1)C(=O)c1ccc(CNC(C)(C)C)cc1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.35
MAPT P10636 1/20 0.34
F10 P00742 1/20 0.34
ALDH1A1 P00352 2/20 0.33
GAA P10253 1/20 0.33
ADRB2 P07550 1/20 0.33
CHRM3 P20309 1/20 0.33
HRH1 P35367 1/20 0.33
DRD3 P35462 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
NAMPT P43490 1/20 0.33
ACHE P22303 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
ADAMTS4 O75173 1/20 0.32
RAB9A P51151 1/20 0.32
USP1 O94782 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695275 0.89 CHRM2 (0.35) CHRM2MAPTALDH1A1GAAADRB2
SCHEMBL4692594 0.84 CHRM2 (0.42) CHRM2ALDH1A1ACHEMEN1KMT2A
SCHEMBL5280124 0.82 CHRM2 (0.46) CHRM2ACHE
SCHEMBL5273742 0.82 NAMPT (0.35) CHRM2MAPTF10DRD3NAMPT
SCHEMBL6021912 0.80 CHRM2 (0.56) CHRM2ALDH1A1ACHERAB9A
SCHEMBL4694973 0.80 MCHR1 (0.40) CHRM2HRH1DRD3HRH3ACHE
SCHEMBL4692420 0.80 MCHR1 (0.38) CHRM2MAPTALDH1A1GAAACHE
SCHEMBL4691377 0.79 KMT2A (0.36) MAPTALDH1A1KMT2ARAB9A
SCHEMBL5807403 0.77 SMYD2 (0.35) CHRM2MAPTALDH1A1CHRM3MEN1
SCHEMBL5273313 0.76 ATR (0.36) MAPTALDH1A1MEN1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893577-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2008-03-05 EP disclosed
WO-2006138218-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-12-28 WO disclosed