SCHEMBL4691377

SCHEMBL4691377

CNCc1ccc(CCC(=O)N(C)CCOC(=O)N(c2ccccc2-c2ccccc2)N2CC[CH]CC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.36
LTB4R2 Q9NPC1 7/20 0.35
LTB4R Q15722 6/20 0.35
FFAR1 O14842 4/20 0.34
FFAR4 Q5NUL3 2/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
HTR7 P34969 1/20 0.33
HTR6 P50406 1/20 0.33
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 3/20 0.31
NPC1 O15118 2/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
PRMT5 O14744 1/20 0.31
WDR77 Q9BQA1 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2639275 0.83 CHRM2 (0.45) KMT2AALDH1A1LMNARAB9ANPC1
SCHEMBL6028157 0.83 ACHE (0.39) LTB4R2HTR1ADRD2HTR7HTR6
SCHEMBL6016864 0.81 BCHE (0.37) HTR1ADRD2HTR7HTR6ALDH1A1
SCHEMBL6022022 0.80 CHRM2 (0.39) HTR1ADRD2HTR7HTR6ALDH1A1
SCHEMBL4695275 0.79 CHRM2 (0.35) KMT2AALDH1A1MAPTCHRNB2CHRNB4
SCHEMBL6022322 0.79 ADRB2 (0.35) ALDH1A1
SCHEMBL4695551 0.77 CNR2 (0.40) KMT2AHTR1ADRD2HTR7HTR6
SCHEMBL4691773 0.76 KDM4E (0.41) KMT2AHTR1ADRD2HTR7HTR6
SCHEMBL6027475 0.76 TRPV1 (0.37) HTR1ADRD2HTR7HTR6LMNA
SCHEMBL5281472 0.76 TAAR1 (0.37) KMT2AALDH1A1L3MBTL1CHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893577-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2008-03-05 EP disclosed
WO-2006138218-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-12-28 WO disclosed