SCHEMBL4696960

SCHEMBL4696960

O=C(O)N1CCc2nn(-c3ccccc3)c(OS(=O)(=O)C(F)(F)F)c2CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 3/20 0.36
GRIA2 P42262 3/20 0.36
SIGMAR1 Q99720 3/20 0.35
ENPP2 Q13822 1/20 0.35
TMEM97 Q5BJF2 2/20 0.35
ADORA1 P30542 1/20 0.35
NTRK1 P04629 2/20 0.34
MGLL Q99685 2/20 0.34
CYP2D6 P10635 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
P2RX7 Q99572 1/20 0.33
LMNA P02545 2/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
ALOX12 P18054 1/20 0.33
FAAH O00519 1/20 0.33
USP2 O75604 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2075004 0.88 GPR119 (0.43) PDK2LMNATHRB
SCHEMBL2075842 0.83 C5AR1 (0.47) PDK2NTRK1
SCHEMBL21893541 0.83 NTRK1 (0.43) PDK2ADORA1NTRK1
SCHEMBL17202496 0.81 F10 (0.38) ADORA1LMNAALDH1A1
SCHEMBL6027740 0.80 CXCR2 (0.32) ADORA1
SCHEMBL2075984 0.79 MEN1 (0.45) PDK2LMNAALDH1A1USP2THRB
SCHEMBL2075003 0.79 TP53 (0.43) LMNA
SCHEMBL2076298 0.79 HPGDS (0.49) LMNA
SCHEMBL2076536 0.78 POLB (0.40) ALDH1A1
SCHEMBL21818847 0.77 P2RX7 (0.37) GRIA2ADORA1CYP2C9P2RX7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1905774-B1 Fused heterocyclic compounds as serotonin receptor modulators JANSSEN PHARMACEUTICA NV (BE) 2013-02-20 EP disclosed
EP-1944306-A1 Fused heterocyclic compounds as serotonin receptor modulators Janssen Pharmaceutica, N.V. (BE) 2008-07-16 EP disclosed
EP-1905774-A1 Fused heterocyclic compounds as serotonin receptor modulators Janssen Pharmaceutica, N.V. (BE) 2008-04-02 EP disclosed