SCHEMBL4698270

SCHEMBL4698270

Cc1ccc([C@H](CC(=O)O)NC(=O)Nc2c(C)ccn(Cc3cccc(F)c3)c2=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CTSA P10619 8/20 0.42
PTGER3 P43115 1/20 0.40
P2RY14 Q15391 1/20 0.40
MAPT P10636 1/20 0.40
ITGB1 P05556 2/20 0.39
ITGA4 P13612 2/20 0.39
LCK P06239 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687794 0.90 MEN1 (0.45) ALDH1A1KDM4ECTSAITGB1ITGA4
SCHEMBL688357 0.84 POLB (0.41) ALDH1A1KDM4ECTSAPTGER3MAPT
SCHEMBL687381 0.84 CTSA (0.47) ALDH1A1KDM4ECTSAPTGER3P2RY14
SCHEMBL687522 0.83 CTSA (0.44) ALDH1A1KDM4ECTSAPTGER3MAPT
SCHEMBL687932 0.82 EGLN1 (0.44) ALDH1A1KDM4ECTSAPTGER3P2RY14
SCHEMBL688110 0.82 MEN1 (0.49) ALDH1A1KDM4ECTSAMAPTITGB1
SCHEMBL687488 0.81 MAPT (0.51) ALDH1A1KDM4ECTSAPTGER3P2RY14
SCHEMBL686919 0.81 GAA (0.45) ALDH1A1KDM4EL3MBTL1CTSAMAPT
SCHEMBL686620 0.80 PTGER3 (0.50) ALDH1A1KDM4ECTSAPTGER3MAPT
SCHEMBL687486 0.80 ALDH1A1 (0.41) ALDH1A1KDM4ECTSAPTGER3ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1176956-B1 CARBOXYLIC ACID DERIVATIVES THAT INHIBIT THE BINDING OF INTEGRINS TO THEIR RECEPTORS ENCYSIVE PHARMACEUTICALS INC (US) 2008-01-09 EP disclosed