SCHEMBL4701221

SCHEMBL4701221

Cc1cc2ccccc2n1Cc1ccc(OCc2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
RAB9A P51151 2/20 0.54
HDAC1 Q13547 1/20 0.53
HDAC2 Q92769 1/20 0.53
HDAC8 Q9BY41 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
HDAC9 Q9UKV0 1/20 0.53
KLK1 P06870 1/20 0.50
KLKB1 P03952 1/20 0.49
TP53 P04637 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
ALOX5 P09917 1/20 0.49
DYRK1A Q13627 3/20 0.48
MAPK1 P28482 1/20 0.48
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2826893 0.87 FFAR1 (0.60) HDAC1HDAC2HDAC8HDAC6HDAC9
SCHEMBL6821030 0.85 HDAC1 (0.62) NPC1MEN1KMT2ARAB9AHDAC1
SCHEMBL30049411 0.85 HDAC1 (0.62) NPC1MEN1KMT2ARAB9AHDAC1
SCHEMBL27204179 0.83 KDM4E (0.58) NPC1MEN1KMT2ARAB9AHDAC1
SCHEMBL4023308 0.81 MTNR1A (0.47) NPC1MEN1KMT2ARAB9AKLKB1
SCHEMBL2825527 0.80 FFAR1 (0.53) HDAC1HDAC2HDAC8HDAC6HDAC9
SCHEMBL5070843 0.80 RAB9A (0.56) NPC1MEN1KMT2ARAB9AHDAC6
SCHEMBL4024812 0.78 CCR2 (0.56) KMT2AKLKB1KDM4EALDH1A1CCR2
SCHEMBL20853225 0.78 HDAC1 (0.62) MEN1KMT2AHDAC1HDAC2HDAC8
SCHEMBL6086266 0.78 HDAC1 (0.62) RAB9AHDAC1HDAC2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951315-A2 PHOSPHOLIPASE INHIBITORS, INCLUDING MULTI-VALENT PHOSPHOLIPASE INHIBITORS, AND USE THEREOF, INCLUDING AS LUMEN-LOCALIZED PHOSPHOLIPASE INHIBITORS Ilypsa, Inc. (US) 2008-08-06 EP disclosed
WO-2007056279-A2 PHOSPHOLIPASE INHIBITORS, INCLUDING MULTI-VALENT PHOSPHOLIPASE INHIBITORS, AND USE THEREOF, INCLUDING AS LUMEN-LOCALIZED PHOSPHOLIPASE INHIBITORS ILYPSA, INC. (US) 2007-05-18 WO disclosed