SCHEMBL4701748

SCHEMBL4701748

CS(=O)(=O)c1cccc(-n2c(-c3ccc(Cl)cc3)nc3c(=O)[nH]c(-c4ccc(-c5cnccn5)cc4)nc32)c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
DHODH Q02127 1/20 0.37
RIPK2 O43353 2/20 0.37
SCD O00767 2/20 0.37
TNKS O95271 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
PSD A5PKW4 2/20 0.36
PTGS2 P35354 1/20 0.35
NR1H2 P55055 2/20 0.34
NR1H3 Q13133 2/20 0.34
AOC3 Q16853 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4701714 0.92 GRM1 (0.40) DHFRALDH1A1HPGDTSHRDHODH
SCHEMBL4699473 0.88 TDP2 (0.45) DHFRALDH1A1HPGDTSHRDHODH
SCHEMBL5612502 0.80 DHFR (0.53) DHFRALDH1A1HPGDTSHRTNKS
SCHEMBL4165879 0.77 RIPK2 (0.40) RIPK2PSDPTGS2AOC3
SCHEMBL4163364 0.77 GRM1 (0.41) TSHRRIPK2PTGS2AOC3
SCHEMBL4169659 0.76 GRM1 (0.58) ALDH1A1HPGDTSHR
SCHEMBL4704624 0.75 TDP2 (0.48) DHFRALDH1A1HPGDTSHRTNKS
SCHEMBL4699312 0.75 TDP2 (0.46) DHFRALDH1A1HPGDTSHRTNKS
SCHEMBL4703457 0.74 GRM1 (0.40) ALDH1A1RIPK2PTGS2AOC3
SCHEMBL5611826 0.73 DHFR (0.49) DHFRALDH1A1HPGDTSHRTNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1999132-A1 AZOLOPYRIMIDINES AS INHIBITORS OF CANNABINOID 1 ACTIVITY IRM, LLC (BM) 2008-12-10 EP disclosed
WO-2007120454-A1 AZOLOPYRIMIDINES AS INHIBITORS OF CANNABINOID 1 ACTIVITY IRM LLC (BM) 2007-10-25 WO disclosed