SCHEMBL4701714

SCHEMBL4701714

NS(=O)(=O)c1cccc(-n2c(-c3ccc(Cl)cc3)nc3c(=O)[nH]c(-c4ccc(-c5cnccn5)cc4)nc32)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 1/20 0.40
DHFR P00374 5/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
CA2 P00918 6/20 0.38
CA9 Q16790 6/20 0.38
CA1 P00915 5/20 0.38
CA12 O43570 4/20 0.38
PTGS2 P35354 1/20 0.36
DHODH Q02127 1/20 0.35
TNKS O95271 2/20 0.35
TNKS2 Q9H2K2 2/20 0.35
PARP2 Q9UGN5 1/20 0.35
PARP1 P09874 1/20 0.35
CHEK2 O96017 1/20 0.35
TDP2 O95551 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4701748 0.92 DHFR (0.38) DHFRALDH1A1HPGDTSHRPTGS2
SCHEMBL4699473 0.85 TDP2 (0.45) DHFRALDH1A1HPGDTSHRDHODH
SCHEMBL4163320 0.77 GRM1 (0.47) GRM1CA2CA9CA1CA12
SCHEMBL4164830 0.76 GRM1 (0.67) GRM1ALDH1A1HPGDTSHR
SCHEMBL4703033 0.74 DHFR (0.39) DHFRALDH1A1HPGDTSHRTNKS
SCHEMBL5611826 0.73 DHFR (0.49) DHFRALDH1A1HPGDTSHRTNKS
SCHEMBL4699926 0.73 DHFR (0.40) DHFRALDH1A1HPGDTSHRTNKS
SCHEMBL5612502 0.73 DHFR (0.53) DHFRALDH1A1HPGDTSHRPTGS2
SCHEMBL4704624 0.72 TDP2 (0.48) DHFRALDH1A1HPGDTSHRPTGS2
SCHEMBL4699312 0.71 TDP2 (0.46) DHFRALDH1A1HPGDTSHRPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1999132-A1 AZOLOPYRIMIDINES AS INHIBITORS OF CANNABINOID 1 ACTIVITY IRM, LLC (BM) 2008-12-10 EP disclosed
WO-2007120454-A1 AZOLOPYRIMIDINES AS INHIBITORS OF CANNABINOID 1 ACTIVITY IRM LLC (BM) 2007-10-25 WO disclosed