SCHEMBL4703202

SCHEMBL4703202

O=C(O)N[C@H]1CCN(C(C(=O)N2CCOCC2)c2cccnc2)C1=O

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
CYP2C9 P11712 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40
F10 P00742 4/20 0.40
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
OXTR P30559 3/20 0.39
F2 P00734 1/20 0.39
KLKB1 P03952 1/20 0.39
P2RX7 Q99572 1/20 0.38
NAMPT P43490 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4702377 0.89 ALDH1A1 (0.55) ALDH1A1CYP3A4CYP2C19F10F2
SCHEMBL8337166 0.86 KDM4D (0.42) ALDH1A1CYP2C9KDM4EHSD17B10F10
SCHEMBL4704111 0.82 ALDH1A1 (0.42) ALDH1A1F10MAPTNAMPT
SCHEMBL4702318 0.78 F10 (0.41) ALDH1A1F10F2KLKB1
SCHEMBL4702226 0.78 F10 (0.71) F10F2KLKB1
SCHEMBL14143923 0.76 ALDH1A1 (0.46) ALDH1A1CYP2C9CYP3A4CYP2C19KDM4E
SCHEMBL4706069 0.75 KDM1A (0.42) F10F2KLKB1
SCHEMBL4495030 0.74 F10 (0.57) F10F2KLKB1
SCHEMBL4706167 0.73 KDM1A (0.51) CYP3A4CYP2C19F10
SCHEMBL6231022 0.73 TACR1 (0.47) ALDH1A1CYP2C9CYP3A4CYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567489-B1 PYRROLIDIN-2-ONE DERIVATIVES AS INHIBITORS OF THROMBIN AND FACTOR XA GLAXO GROUP LTD (GB) 2008-07-23 EP disclosed