SCHEMBL4703530

SCHEMBL4703530

CCn1cc(N(C)C(=O)n2ccc([N+](=O)[O-])c2)cc1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 8/20 0.40
ATM Q13315 1/20 0.36
ALDH1A1 P00352 4/20 0.36
TP53 P04637 1/20 0.36
HTT P42858 1/20 0.36
HCAR3 P49019 1/20 0.34
KEAP1 Q14145 2/20 0.34
NFE2L2 Q16236 2/20 0.34
HTR7 P34969 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4701014 0.87 AR (0.51) ARATMALDH1A1
SCHEMBL8393115 0.84 AR (0.48) ARATMALDH1A1
SCHEMBL4703944 0.75 HTT (0.40) ARALDH1A1TP53HTTMAPT
SCHEMBL883063 0.71 MAPK1 (0.43) ARALDH1A1TP53HTTSMN1; SMN2
SCHEMBL7838764 0.70 SMN1; SMN2 (0.34) ATMALDH1A1MAPTSMN1; SMN2
SCHEMBL8388682 0.68 MMP14 (0.34) MAPT
SCHEMBL6800421 0.67 TDP1 (0.44) ALDH1A1TP53
SCHEMBL5676062 0.65 AR (0.41) ARALDH1A1TP53HTTMAPT
SCHEMBL7056737 0.65 ALDH1A1 (0.34) ARALDH1A1TP53HTTHCAR3
SCHEMBL5680368 0.64 AR (0.38) ARALDH1A1TP53HTTKEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678133-A4 SEQUENCE SELECTIVE PYRROLE AND IMIDAZOLE POLYAMIDE METALLOCOMPLEXES UNIV WESTERN SYDNEY (AU) 2008-06-18 EP disclosed
EP-1678133-A1 SEQUENCE SELECTIVE PYRROLE AND IMIDAZOLE POLYAMIDE METALLOCOMPLEXES University of Western Sydney (AU) 2006-07-12 EP disclosed
WO-2005033077-A1 SEQUENCE SELECTIVE PYRROLE AND IMIDAZOLE POLYAMIDE METALLOCOMPLEXES UNIVERSITY OF WESTERN SYDNEY (AU) 2005-04-14 WO disclosed