SCHEMBL4704282

SCHEMBL4704282

CC(C)(C)N(C(=O)O)[C@@H](Cc1ccncc1)C(=O)N1CCOCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.44
TSHR P16473 2/20 0.44
MMP8 P22894 1/20 0.42
NAMPT P43490 1/20 0.38
POLB P06746 1/20 0.38
KDM4E B2RXH2 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
LMNA P02545 2/20 0.37
HSD17B10 Q99714 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ALDH1A1 P00352 3/20 0.36
TACR1 P25103 2/20 0.36
MME P08473 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
CAMK2D Q13557 1/20 0.36
P2RX4 Q99571 1/20 0.36
P2RX7 Q99572 1/20 0.36
CAMK2A Q9UQM7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15153143 0.90 CHRM1 (0.46) CHRM1TSHRKDM4ESMN1; SMN2LMNA
SCHEMBL15153161 0.90 CHRM1 (0.46) CHRM1TSHRKDM4ESMN1; SMN2LMNA
SCHEMBL4704760 0.87 CHRM1 (0.48) CHRM1TSHRMMP8POLBLMNA
SCHEMBL4705390 0.86 TSHR (0.46) TSHRMMP8SMN1; SMN2NPC1RAB9A
SCHEMBL1312285 0.80 MMP8 (0.50) CHRM1TSHRMMP8KDM4EHSD17B10
Hydrochloric Acid SCHEMBL1311367 0.79 MMP8 (0.49) CHRM1TSHRMMP8KDM4EHSD17B10
SCHEMBL7708347 0.79 KLKB1 (0.41)
SCHEMBL4702059 0.78 OPRD1 (0.41) TSHRALDH1A1HTT
SCHEMBL3738889 0.78 CTSD (0.40) TSHRPOLBSMN1; SMN2ALDH1A1TACR1
SCHEMBL3450371 0.77 F10 (0.42) CHRM1TSHRKDM4ESMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567489-B1 PYRROLIDIN-2-ONE DERIVATIVES AS INHIBITORS OF THROMBIN AND FACTOR XA GLAXO GROUP LTD (GB) 2008-07-23 EP disclosed