SCHEMBL4705384

SCHEMBL4705384

N#Cc1ccccc1C(=O)c1ccccc1-c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.39
ALDH1A1 P00352 2/20 0.38
GAA P10253 1/20 0.38
PTGER4 P35408 2/20 0.37
IDO1 P14902 3/20 0.36
TDO2 P48775 3/20 0.36
TSHR P16473 1/20 0.36
RORC P51449 2/20 0.35
RORB Q92753 1/20 0.35
CDC7 O00311 2/20 0.35
PLK4 O00444 1/20 0.35
AURKA O14965 1/20 0.35
MAPK13 O15264 1/20 0.35
DAPK3 O43293 1/20 0.35
ROCK2 O75116 1/20 0.35
RPS6KA5 O75582 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
PRKCG P05129 1/20 0.35
CDK1 P06493 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707011 0.87 IDO1 (0.44) TACR1ALDH1A1GAAPTGER4IDO1
SCHEMBL4757295 0.86 RORB (0.51) TACR1ALDH1A1GAAPTGER4IDO1
SCHEMBL4708172 0.80 RORB (0.46) TACR1RORCRORBCDC7MAPK1
SCHEMBL4707863 0.75 IDH1 (0.44) TACR1RORCRORBGPBAR1
SCHEMBL4638919 0.75 TACR1 (0.48) TACR1ALDH1A1GAATSHRRORC
SCHEMBL4707172 0.75 RORB (0.46) ALDH1A1GAAPTGER4TSHRRORC
SCHEMBL4706420 0.75 IDO1 (0.44) TACR1PTGER4IDO1TDO2CDC7
SCHEMBL4708046 0.75 RORB (0.42) TACR1RORCRORBGPBAR1
SCHEMBL4707969 0.75 CDC7 (0.42) TACR1ALDH1A1GAARORCRORB
SCHEMBL4707650 0.74 RORB (0.41) ALDH1A1GAAPTGER4TSHRRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed