SCHEMBL4705631

SCHEMBL4705631

CC(C)(C)[Si](C)(C)OCC#CC(=O)c1ccccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
ERCC5 P28715 1/20 0.36
FEN1 P39748 1/20 0.36
ALDH1A1 P00352 4/20 0.36
POLB P06746 1/20 0.34
RAB9A P51151 3/20 0.34
KMT2A Q03164 2/20 0.34
LMNA P02545 2/20 0.34
JAK2 O60674 1/20 0.34
TYK2 P29597 1/20 0.34
HTT P42858 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
NPC1 O15118 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4706996 0.83 ALDH1A1 (0.36) ALDH1A1RAB9AKMT2ALMNAKDM4E
SCHEMBL974627 0.81 BACE1 (0.37) ADRB2ADRB1ADRB3CES1ALDH1A1
SCHEMBL8017463 0.79 ERCC5 (0.44) ADRB2ADRB1ADRB3CES2CES1
SCHEMBL28100608 0.74 CES2 (0.48) CES2CES1ERCC5FEN1ALDH1A1
SCHEMBL20089301 0.73 DGAT1 (0.30)
SCHEMBL19520131 0.73 KDM4E (0.34) ALDH1A1POLBKMT2AHTTKDM4E
SCHEMBL4708420 0.72 CES2 (0.41) ADRB2ADRB1ADRB3CES2CES1
SCHEMBL7402519 0.72 NPSR1 (0.35) ALDH1A1POLBRAB9AKMT2AHTT
SCHEMBL10717928 0.71 ERCC5 (0.44) CES2CES1ERCC5FEN1ALDH1A1
SCHEMBL11033388 0.70 CES2 (0.48) CES2CES1ERCC5FEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed