SCHEMBL4705960

SCHEMBL4705960

CCCC[Sn](CCCC)(CCCC)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1cncnc1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
POLB P06746 1/20 0.33
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31
HTT P42858 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CYP1A2 P05177 1/20 0.31
METAP2 P50579 1/20 0.31
GABRA2 P47869 1/20 0.30
GABRB2 P47870 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4759295 0.88 POLB (0.37) HSP90AA1HSP90AB1POLBGRIN1GRIN2B
SCHEMBL4706975 0.88 HSP90AA1 (0.35) HSP90AA1HSP90AB1POLBGRIN1GRIN2B
SCHEMBL4638838 0.86 POLB (0.38) HSP90AA1HSP90AB1POLBHTTL3MBTL1
SCHEMBL4707593 0.83 P2RX7 (0.36) HSP90AA1HSP90AB1GABRA2GABRB2
SCHEMBL4707683 0.81 HSP90AA1 (0.35) HSP90AA1HSP90AB1POLBHTTL3MBTL1
SCHEMBL4708507 0.79 HSP90AA1 (0.34) HSP90AA1HSP90AB1POLBL3MBTL1CYP1A2
SCHEMBL4708592 0.78 HSP90AA1 (0.33) HSP90AA1HSP90AB1POLBGABRA2GABRB2
SCHEMBL4708607 0.77 GABRA2 (0.35) HSP90AA1HSP90AB1GABRA2GABRB2
SCHEMBL3673183 0.76 CDC7 (0.48)
SCHEMBL4804309 0.73 PAX8 (0.35) HSP90AA1HSP90AB1POLBGABRA2GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed