SCHEMBL4708607

SCHEMBL4708607

CCCC[Sn](CCCC)(CCCC)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1C1CC1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GABRA2 P47869 4/20 0.35
GABRB2 P47870 4/20 0.35
PDE8B O95263 1/20 0.34
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
JAK3 P52333 1/20 0.33
DPP4 P27487 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
GRM2 Q14416 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.30
PTGER4 P35408 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707683 0.83 HSP90AA1 (0.35) GABRA2GABRB2HSP90AA1HSP90AB1
SCHEMBL3667322 0.81 ROCK2 (0.43) JAK2GRM2
SCHEMBL4708592 0.80 HSP90AA1 (0.33) GABRA2GABRB2HSP90AA1HSP90AB1PTGER4
SCHEMBL4638838 0.77 POLB (0.38) HSP90AA1HSP90AB1GRM2PTGER4
SCHEMBL4804309 0.77 PAX8 (0.35) GABRA2GABRB2JAK2JAK1JAK3
SCHEMBL4706975 0.77 HSP90AA1 (0.35) GABRA2GABRB2HSP90AA1HSP90AB1GRM2
SCHEMBL4705960 0.77 HSP90AA1 (0.33) GABRA2GABRB2HSP90AA1HSP90AB1
SCHEMBL4297826 0.76 CDC7 (0.44) JAK2
SCHEMBL4708507 0.74 HSP90AA1 (0.34) HSP90AA1HSP90AB1GRM2
SCHEMBL4707593 0.74 P2RX7 (0.36) GABRA2GABRB2HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed