SCHEMBL4707136

SCHEMBL4707136

COc1ccccc1C(=O)c1cccnc1Br

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.51
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
NPC1 O15118 3/20 0.51
TP53 P04637 1/20 0.51
GAA P10253 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
CNR2 P34972 1/20 0.48
CTSD P07339 1/20 0.45
HSD17B10 Q99714 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
CDK5 Q00535 1/20 0.44
CDK5R1 Q15078 1/20 0.44
POLB P06746 1/20 0.44
LMNA P02545 1/20 0.44
ALOX15 P16050 1/20 0.44
RXFP1 Q9HBX9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12205524 0.83 RAB9A (0.52) RAB9AMEN1KMT2ANPC1TP53
SCHEMBL1643645 0.82 LMNA (0.46) RAB9AMEN1KMT2ANPC1TP53
SCHEMBL10899012 0.81 RAB9A (0.56) RAB9AMEN1KMT2ANPC1TP53
SCHEMBL322168 0.81 CTSD (0.62) RAB9ANPC1SMN1; SMN2CNR2CTSD
SCHEMBL29658169 0.81 CTSD (0.62) RAB9ANPC1SMN1; SMN2CNR2CTSD
SCHEMBL27789892 0.79 CTSD (0.60) RAB9ANPC1SMN1; SMN2CNR2CTSD
SCHEMBL4706785 0.79 CTNNB1 (0.46) RAB9AKMT2ANPC1TP53SMN1; SMN2
SCHEMBL9575507 0.78 CTSD (0.51) RAB9ANPC1GAASMN1; SMN2CNR2
SCHEMBL7496703 0.78 RAB9A (0.51) RAB9AMEN1KMT2ANPC1TP53
SCHEMBL30118936 0.78 RAB9A (0.71) RAB9AMEN1KMT2ANPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed
CN-1646502-A Triazole derivatives as tachykinin receptor antagonists LILLY CO ELI (US) 2005-07-27 CN disclosed