SCHEMBL4706785

SCHEMBL4706785

Cc1ccccc1C(=O)c1cccnc1Br

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 1/20 0.46
WNT3A P56704 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
KMT2A Q03164 1/20 0.45
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
TP53 P04637 1/20 0.43
MAPK1 P28482 1/20 0.43
ELANE P08246 2/20 0.42
PLAU P00749 1/20 0.42
MYC P01106 1/20 0.41
TYK2 P29597 1/20 0.41
KDM4E B2RXH2 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ENPP3 O14638 1/20 0.41
ALPL P05186 1/20 0.41
XIAP P98170 1/20 0.41
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705926 0.79 CES2 (0.47) CTNNB1WNT3AL3MBTL1KMT2ANPC1
SCHEMBL29896666 0.79 CES2 (0.47) CTNNB1WNT3AL3MBTL1KMT2ANPC1
SCHEMBL2901555 0.79 RORB (0.55) KMT2ASMN1; SMN2ALDH1A1
SCHEMBL29387256 0.79 CYP3A4 (0.55) KMT2ATP53SMN1; SMN2ALDH1A1ENPP3
SCHEMBL333141 0.79 CYP3A4 (0.55) KMT2ATP53SMN1; SMN2ALDH1A1ENPP3
SCHEMBL4707136 0.79 RAB9A (0.51) KMT2ANPC1RAB9ATP53KDM4E
SCHEMBL4707275 0.79 AKR1C3 (0.52) L3MBTL1KMT2ANPC1RAB9AKDM4E
SCHEMBL7851627 0.78 KDM4E (0.62) CTNNB1WNT3AL3MBTL1KMT2AMYC
SCHEMBL8764829 0.77 CTNNB1 (0.44) CTNNB1WNT3AL3MBTL1KMT2ANPC1
SCHEMBL8691222 0.77 L3MBTL1 (0.54) CTNNB1WNT3AL3MBTL1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed
CN-1312136-C Triazole derivatives as tachykinin receptor antagonists LILLY CO ELI (US) 2007-04-25 CN disclosed
CN-1646502-A Triazole derivatives as tachykinin receptor antagonists LILLY CO ELI (US) 2005-07-27 CN disclosed