SCHEMBL4707331

SCHEMBL4707331

Cc1cc(Cc2ccccc2Cl)c(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2-c2cccnc2)nn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.37
P2RX7 Q99572 7/20 0.36
GRM2 Q14416 1/20 0.35
POLB P06746 1/20 0.34
HTT P42858 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
ALDH1A1 P00352 1/20 0.33
TRPA1 O75762 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
GRIN2B Q13224 1/20 0.32
CDC7 O00311 1/20 0.32
MAP4K4 O95819 1/20 0.32
PIM1 P11309 1/20 0.32
PRKACA P17612 1/20 0.32
CDK2 P24941 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708132 0.91 GRM2 (0.36) P2RX7GRM2POLBHTTL3MBTL1
SCHEMBL4707706 0.83 IDH1 (0.42) IDH1P2RX7GPBAR1
SCHEMBL4707319 0.81 GRM2 (0.36) P2RX7GRM2HTTL3MBTL1SMN1; SMN2
SCHEMBL4708438 0.80 CDC7 (0.41) GRM2HTTL3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL5633626 0.76 IDH1 (0.42) IDH1P2RX7GRM2POLBHTT
SCHEMBL4706229 0.76 IDH1 (0.44) IDH1GRM2NPC1RAB9ASMN1; SMN2
SCHEMBL6388287 0.76 IDH1 (0.39) IDH1P2RX7GRM2NPC1RAB9A
SCHEMBL4705841 0.76 IDH1 (0.36) IDH1P2RX7GRM2POLBHTT
SCHEMBL4709676 0.75 RORB (0.46) IDH1
SCHEMBL4707893 0.75 P2RX7 (0.41) IDH1P2RX7GRM2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed