SCHEMBL4705841

SCHEMBL4705841

Cc1nnc(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2-c2cccnc2)n1[C@H](C)c1ccccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.36
P2RX7 Q99572 5/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
GRM2 Q14416 1/20 0.34
CDC7 O00311 3/20 0.34
MAP4K4 O95819 2/20 0.33
PIM1 P11309 2/20 0.33
PRKACA P17612 2/20 0.33
CDK2 P24941 2/20 0.33
GSK3B P49841 2/20 0.33
HIPK2 Q9H2X6 2/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
POLB P06746 1/20 0.33
DAPK3 O43293 1/20 0.33
ROCK2 O75116 1/20 0.33
PRKD3 O94806 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707918 0.91 CDC7 (0.38) P2RX7GRM2CDC7MAP4K4PIM1
SCHEMBL4705551 0.80 CDC7 (0.42) CDC7MAP4K4PIM1PRKACACDK2
SCHEMBL4707828 0.80 CDC7 (0.42) CDC7MAP4K4PIM1PRKACACDK2
SCHEMBL6388287 0.80 IDH1 (0.39) IDH1P2RX7NPC1RAB9ASMN1; SMN2
SCHEMBL4708876 0.79 GHSR (0.38) SMN1; SMN2HTT
SCHEMBL4705055 0.78 ALDH1A1 (0.34) SMN1; SMN2CDC7HTTL3MBTL1
SCHEMBL4707331 0.76 IDH1 (0.37) IDH1P2RX7NPC1RAB9ASMN1; SMN2
SCHEMBL4707548 0.75 CDC7 (0.40) GRM2CDC7MAP4K4PIM1PRKACA
SCHEMBL5633626 0.75 IDH1 (0.42) IDH1P2RX7NPC1RAB9ASMN1; SMN2
SCHEMBL4705321 0.74 TACR1 (0.35) SMN1; SMN2GRM2CDC7MAP4K4PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed