SCHEMBL4707918

SCHEMBL4707918

Cc1nnc(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2-c2ccncc2)n1[C@H](C)c1ccccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 6/20 0.38
MAP4K4 O95819 5/20 0.36
PRKACA P17612 5/20 0.36
CDK2 P24941 5/20 0.36
GSK3B P49841 5/20 0.36
ROCK2 O75116 4/20 0.36
DAPK3 O43293 3/20 0.36
PRKD3 O94806 3/20 0.36
FLT3 P36888 3/20 0.36
CLK2 P49760 3/20 0.36
PRKX P51817 3/20 0.36
JAK3 P52333 3/20 0.36
CDK5 Q00535 3/20 0.36
MAP4K2 Q12851 3/20 0.36
CAMK2D Q13557 3/20 0.36
DYRK1A Q13627 3/20 0.36
PKN2 Q16513 3/20 0.36
STK17A Q9UEE5 3/20 0.36
MAP4K5 Q9Y4K4 3/20 0.36
PIM1 P11309 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705841 0.91 IDH1 (0.36) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4705321 0.83 TACR1 (0.35) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4707828 0.82 CDC7 (0.42) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4705551 0.82 CDC7 (0.42) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4707454 0.82 CDC7 (0.38) CDC7MAP4K4PRKACACDK2GSK3B
SCHEMBL4708876 0.81 GHSR (0.38) HTTTACR1
SCHEMBL4705055 0.80 ALDH1A1 (0.34) CDC7MAPK13MAPK12MAPK9HTT
SCHEMBL4705363 0.78 GRM2 (0.36) CDC7GRM2PTGER4HSP90AA1HSP90B1
SCHEMBL14279238 0.78 GRM2 (0.36) CDC7GRM2PTGER4HSP90AA1HSP90B1
SCHEMBL4707457 0.77 CDC7 (0.42) CDC7MAP4K4PRKACACDK2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed