SCHEMBL4707992

SCHEMBL4707992

CC(OC(C)(C)C)c1onc(-c2nnn(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2Cl)c1C(=O)c1ccccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 8/20 0.36
RORB Q92753 5/20 0.35
RORC P51449 3/20 0.35
TACR1 P25103 1/20 0.34
AKR1C3 P42330 2/20 0.34
KMT2A Q03164 1/20 0.34
NR1H4 Q96RI1 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SLC16A3 O15427 1/20 0.32
SLC16A1 P53985 1/20 0.32
MCTS1 Q9ULC4 1/20 0.32
AKR1C2 P52895 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707988 1.00 PTGER4 (0.36) PTGER4RORBRORCTACR1AKR1C3
SCHEMBL4708475 0.90 RORB (0.37) PTGER4RORBRORCTACR1AKR1C3
SCHEMBL4708474 0.90 RORB (0.37) PTGER4RORBRORCTACR1AKR1C3
SCHEMBL4705104 0.88 POLB (0.35) PTGER4KMT2AKDM4ESMN1; SMN2
SCHEMBL4637886 0.85 EPAS1 (0.39) PTGER4TACR1KMT2ANR1H4KDM4E
SCHEMBL4705694 0.85 LMNA (0.43) RORBRORCTACR1KMT2A
SCHEMBL4708267 0.83 RORB (0.38) RORBRORCTACR1AKR1C3KMT2A
SCHEMBL4638837 0.78 ALDH1A1 (0.38) TACR1KMT2ANR1H4HTTSMN1; SMN2
SCHEMBL4707456 0.78 POLB (0.37) RORCTACR1KMT2AKDM4ESMN1; SMN2
SCHEMBL4707455 0.78 POLB (0.37) RORCTACR1KMT2AKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed