SCHEMBL4708299

SCHEMBL4708299

COc1ccccc1C(O)c1cccnc1Br

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.49
ACHE P22303 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
PLAU P00749 1/20 0.41
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM5 P08912 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
CTSA P10619 1/20 0.38
LMNA P02545 2/20 0.38
AGTR1 P30556 1/20 0.38
CYP1A2 P05177 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ATM Q13315 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL238441 0.80 CA1 (0.57) TDP1ACHESMN1; SMN2ALDH1A1MAPT
SCHEMBL4706914 0.80 GAA (0.53) MAPTPLAUCTSAKDM4EL3MBTL1
SCHEMBL24631622 0.78 CHRM2 (0.45) TDP1ACHESMN1; SMN2CHRM2CHRM4
SCHEMBL4707217 0.77 CYP2C19 (0.45) TDP1SMN1; SMN2ALDH1A1MAPTCTSA
SCHEMBL4708317 0.77 HDAC4 (0.40) MAPTCTSALMNAKDM4ETP53
SCHEMBL11398150 0.77 ACHE (0.51) TDP1ACHESMN1; SMN2ALDH1A1MAPT
SCHEMBL162184 0.77
SCHEMBL30454545 0.77
SCHEMBL4706109 0.76 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1MAPTLMNAMEN1
Ammonia Solution, Strong SCHEMBL28240370 0.75 PLAU (0.46) SMN1; SMN2PLAULMNACYP1A2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed
CN-1646502-A Triazole derivatives as tachykinin receptor antagonists LILLY CO ELI (US) 2005-07-27 CN disclosed