SCHEMBL4711347

SCHEMBL4711347

CNC(=O)C1(c2ccc(O)cc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 3/20 0.42
OPRL1 P41146 1/20 0.42
APP P05067 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP3A4 P08684 1/20 0.41
ESR1 P03372 2/20 0.41
ESR2 Q92731 2/20 0.41
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
P2RX7 Q99572 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
LMNA P02545 3/20 0.38
HSD11B1 P28845 3/20 0.38
PKM P14618 1/20 0.37
HDAC1 Q13547 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CFTR P13569 1/20 0.37
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22027296 0.91 HDAC4 (0.51) HDAC4ESR1ESR2ALDH1A1SMN1; SMN2
SCHEMBL25975348 0.85 MAPT (0.48) HDAC4OPRL1CYP2C19CYP3A4ALDH1A1
SCHEMBL3553242 0.83 HDAC4 (0.62) HDAC4ALDH1A1SMN1; SMN2LMNAHSD11B1
SCHEMBL8572144 0.82 HDAC4 (0.59) HDAC4OPRL1ALDH1A1SMN1; SMN2P2RX7
SCHEMBL4711696 0.80 ALDH1A1 (0.59) CYP2C19CYP3A4ALDH1A1SMN1; SMN2CYP2C9
SCHEMBL19537445 0.79 LMNA (0.50) HDAC4OPRL1ALDH1A1LMNAHSD11B1
SCHEMBL12120029 0.78 ESR2 (0.45) APPCYP2C19CYP3A4ESR1ESR2
SCHEMBL1335906 0.77 ESR2 (0.48) HDAC4APPCYP2C19CYP3A4ESR1
SCHEMBL1464894 0.77 CA12 (0.44) APPCYP2C19CYP3A4ESR1ESR2
SCHEMBL25460818 0.77 HDAC4 (0.73) HDAC4ALDH1A1SMN1; SMN2LMNAHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025050125-A1 SUBSTITUTED BENZOXAZOLYLAMINO BENZOXAZOLES IMMVENTION THERAPEUTIX (US) 2025-03-06 WO disclosed
EP-1660504-B1 THIENOPYRIDINE-PHENYLACET AMIDES AND THEIR DERIVATIVES USEFUL AS NEW ANTI-ANGIOGENIC AGENTS PFIZER (US) 2008-10-29 EP disclosed
EP-1660504-B1 THIENOPYRIDINE-PHENYLACET AMIDES AND THEIR DERIVATIVES USEFUL AS NEW ANTI-ANGIOGENIC AGENTS PFIZER (US) 2008-10-29 EP disclosed
US-7208500-B2 Thienopyridine-phenylacetamides and their derivatives useful as new anti-angiogenic agents AGOURON PHARMACEUTICALS, INC. (US) 2007-04-24 US disclosed
US-7208500-B2 Thienopyridine-phenylacetamides and their derivatives useful as new anti-angiogenic agents AGOURON PHARMACEUTICALS, INC. (US) 2007-04-24 US disclosed
US-7208500-B2 Thienopyridine-phenylacetamides and their derivatives useful as new anti-angiogenic agents AGOURON PHARMACEUTICALS, INC. (US) 2007-04-24 US disclosed
EP-1660504-A1 THIENOPYRIDINE-PHENYLACET AMIDES AND THEIR DERIVATIVES USEFUL AS NEW ANTI-ANGIOGENIC AGENTS PFIZER INC. (US) 2006-05-31 EP disclosed
US-20050090509-A1 Thienopyridine-phenylacetamides and their derivatives useful as new anti-angiogenic agents Agouron Pharmaceuticals,Inc. 2005-04-28 US disclosed
WO-2005021554-A1 THIENOPYRIDINE-PHENYLACET AMIDES AND THEIR DERIVATIVES USEFUL AS NEW ANTI-ANGIOGENIC AGENTS PFIZER INC. (US) 2005-03-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050090509-A1 Thienopyridine-phenylacetamides and their derivatives useful as new anti-angiogenic agents CCNA1, PGF, CCNA2 HDAC4 1249/4885OPRL1 2495/4885APP 3683/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.