SCHEMBL4712463

SCHEMBL4712463

Cc1cccc(C#Cc2cccc(-n3cnc(C(=O)O)n3)c2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
KDM4E B2RXH2 1/20 0.49
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
PKM P14618 1/20 0.49
HPGD P15428 1/20 0.49
ALOX15 P16050 1/20 0.49
CYP2C19 P33261 1/20 0.49
THPO P40225 1/20 0.49
KMT2A Q03164 1/20 0.49
GRIN2B Q13224 1/20 0.49
GRM1 Q13255 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4711597 0.88 GRM5 (0.44) GRM5NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL4713592 0.86 GRM5 (0.44) GRM5
SCHEMBL4711486 0.84 GRM5 (0.46) GRM5NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL4711268 0.79 GRM5 (0.43) GRM5NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL4713871 0.79 GRM5 (0.42) GRM5
SCHEMBL20594437 0.77 GRM5 (0.54) GRM5SMN1; SMN2ALDH1A1TP53
SCHEMBL29794847 0.77 GRM5 (0.54) GRM5SMN1; SMN2ALDH1A1TP53
SCHEMBL15020092 0.75 MEN1 (0.55) NPC1SMN1; SMN2MEN1ALDH1A1TP53
SCHEMBL4710432 0.74 GRM5 (0.53) GRM5NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL15019823 0.71 MAPT (0.50) SMN1; SMN2KDM4EALDH1A1TP53PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0998459-B1 PYRIDINE DERIVATIVES NOVARTIS AG (CH) 2008-04-23 EP claimed