SCHEMBL4715365

SCHEMBL4715365

CN(CCc1ccc(F)cc1)C1CN(C(=O)O)C1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 8/20 0.47
TAAR1 Q96RJ0 1/20 0.46
AOC3 Q16853 1/20 0.44
CHRM1 P11229 4/20 0.43
CHRM5 P08912 3/20 0.43
CHRM3 P20309 3/20 0.43
CYP2D6 P10635 1/20 0.43
HRH1 P35367 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
MCHR1 Q99705 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4715512 0.82 SLC6A4 (0.48) L3MBTL1MCHR1CHRM4
SCHEMBL4714391 0.81 SMN1; SMN2 (0.44) CYP2D6L3MBTL1
SCHEMBL1969047 0.77 TAAR1 (0.60) TAAR1AOC3CHRM1CYP2D6HRH1
SCHEMBL4711078 0.75 L3MBTL1 (0.42) AGTR2TAAR1L3MBTL1
SCHEMBL29056938 0.75 L3MBTL1 (0.66) AGTR2CYP2D6L3MBTL1SIGMAR1
SCHEMBL27544931 0.73 CHIA (0.52) AGTR2TAAR1CHRM1CHRM3CYP2D6
SCHEMBL4713293 0.73 TAAR1 (0.49) AGTR2TAAR1AOC3L3MBTL1SIGMAR1
Oxalic Acid SCHEMBL7470413 0.72 KMT2A (0.57) CHRM1CYP2D6HRH1L3MBTL1MCHR1
SCHEMBL28550033 0.72 HRH3 (0.35) L3MBTL1
SCHEMBL144125 0.72 KMT2A (0.51) AGTR2SIGMAR1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1933830-A1 ANTAGONISTS OF SNS SODIUM CHANNELS Vernalis (R&D) Limited (GB) 2008-06-25 EP disclosed
WO-2007007057-A1 ANTAGONISTS OF SNS SODIUM CHANNELS VERNALIS (R & D) LIMITED (GB) 2007-01-18 WO disclosed