SCHEMBL4713293

SCHEMBL4713293

CN(CCc1ccccc1Cl)C1CN(C(=O)O)C1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.49
AOC3 Q16853 1/20 0.47
CCR5 P51681 1/20 0.42
MGLL Q99685 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HTR2A P28223 1/20 0.39
AGTR2 P50052 2/20 0.38
SIGMAR1 Q99720 1/20 0.38
MBTPS1 Q14703 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4711078 0.86 L3MBTL1 (0.42) TAAR1L3MBTL1HTR2AAGTR2MBTPS1
SCHEMBL4714391 0.84 SMN1; SMN2 (0.44) SLC6A2SLC6A4L3MBTL1
SCHEMBL27817763 0.78 TAAR1 (0.62) TAAR1AOC3SLC6A2SLC6A4HTR2A
SCHEMBL22462903 0.76 KCNH2 (0.41) TAAR1
SCHEMBL4695317 0.73 KCNH2 (0.53) CCR5HTR2A
SCHEMBL4715365 0.73 AGTR2 (0.47) TAAR1AOC3L3MBTL1AGTR2SIGMAR1
SCHEMBL144125 0.73 KMT2A (0.51) AGTR2SIGMAR1
SCHEMBL18422574 0.72 TAAR1 (0.62) TAAR1AOC3SLC6A2SLC6A4
SCHEMBL17274372 0.71 NAAA (0.63) TAAR1CCR5
SCHEMBL18567998 0.71 MBTPS1 (0.51) TAAR1AOC3SLC6A2SLC6A4MBTPS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1933830-A1 ANTAGONISTS OF SNS SODIUM CHANNELS Vernalis (R&D) Limited (GB) 2008-06-25 EP disclosed
WO-2007007057-A1 ANTAGONISTS OF SNS SODIUM CHANNELS VERNALIS (R & D) LIMITED (GB) 2007-01-18 WO disclosed