SCHEMBL4715466

SCHEMBL4715466

CS(=O)(=O)c1cccc(-c2ccc3[nH]c(=O)c4[nH]ccc4c3c2)c1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FASN P49327 1/20 0.45
PDPK1 O15530 1/20 0.44
PTGS2 P35354 7/20 0.41
CAMKK2 Q96RR4 2/20 0.39
TTK P33981 1/20 0.39
SCD O00767 4/20 0.38
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
MAP3K5 Q99683 1/20 0.38
PLK4 O00444 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Propionic Acid SCHEMBL4155344 0.92 FASN (0.42) FASNPDPK1PTGS2CAMKK2TTK
Butyric Acid SCHEMBL4153848 0.90 FASN (0.41) FASNPDPK1PTGS2CAMKK2TTK
3-Methylbutanoic Acid SCHEMBL4163003 0.88 FASN (0.40) FASNPDPK1PTGS2CAMKK2NR1H2
SCHEMBL4159560 0.87 VCP (0.41) FASNPDPK1PTGS2CAMKK2
Propionic Acid SCHEMBL4155190 0.81 PTGS2 (0.40) PTGS2
SCHEMBL4713436 0.80 PARP1 (0.46) PDPK1
Propionic Acid SCHEMBL4159324 0.77 FASN (0.48) FASNCAMKK2
SCHEMBL3242761 0.77 CAMKK2 (0.46) FASNPDPK1PTGS2CAMKK2
Propionic Acid SCHEMBL4153840 0.77 PIM1 (0.44)
SCHEMBL13951195 0.77 PDPK1 (0.38) FASNPDPK1PTGS2CAMKK2MAP3K5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-A1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PIERRE FABRE MEDICAMENT (FR) 2008-03-19 EP disclosed
WO-2007003611-A1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PIERRE FABRE MEDICAMENT (FR) 2007-01-11 WO disclosed