SCHEMBL4715540

SCHEMBL4715540

Cc1cccc(CCNC2CN(C(=O)O)C2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
AKR1C3 P42330 1/20 0.44
POLB P06746 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CNR1 P21554 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 2/20 0.43
TACR1 P25103 1/20 0.43
BCHE P06276 1/20 0.43
CTDSP1 Q9GZU7 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4713692 0.83 TAAR1 (0.44) NPC1RAB9APOLBTAAR1KMT2A
SCHEMBL4716650 0.76 TP53 (0.42) NPC1RAB9APOLBTAAR1MEN1
SCHEMBL29101911 0.75 TAAR1 (0.44) NPC1TAAR1CNR1DRD4
SCHEMBL4713876 0.75 TLR2 (0.50) TAAR1MEN1KMT2ATDP1ALDH1A1
SCHEMBL11895626 0.74 NPC1 (0.65) NPC1RAB9AAKR1C3POLBTAAR1
SCHEMBL15054786 0.72 TAAR1 (0.66) NPC1RAB9ATAAR1MEN1KMT2A
SCHEMBL4342706 0.72 TAAR1 (0.66) NPC1RAB9ATAAR1MEN1KMT2A
SCHEMBL3316633 0.70 SLC6A9 (0.44) MEN1KMT2AGAA
SCHEMBL10112805 0.69 HDAC3 (0.59) NPC1RAB9APOLBHDAC3HDAC1
SCHEMBL3213481 0.69 HDAC3 (0.52) NPC1RAB9AAKR1C3POLBTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1933830-A1 ANTAGONISTS OF SNS SODIUM CHANNELS Vernalis (R&D) Limited (GB) 2008-06-25 EP disclosed
WO-2007007057-A1 ANTAGONISTS OF SNS SODIUM CHANNELS VERNALIS (R & D) LIMITED (GB) 2007-01-18 WO disclosed